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Home > Products > APIs cancer> Hot APIs cancer> PD-166285 dihydrochloride;PD-166285 2HCl;PD166285 dihydrochloride,CAS212391-63-4
PD-166285 dihydrochloride;PD-166285 2HCl;PD166285 dihydrochloride,CAS212391-63-4
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R-SX-1304 1 ¥ 1
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分子量 585.35
溶解度 N/A
CAS號 212391-63-4
質(zhì)量控制 N/A
儲存條件 N/A
保存時間 N/A
其他信息 價格1,就是價格現(xiàn)詢
PD 166285, a novel protein tyrosine kinase inhibitor of a new structural class, is a potent inhibitor of the tyrosine kinases c-Src, Flg (fibroblast growth factor receptor 1, FGFR1), and PDGFRβ (platelet-derived growth factor receptor β) (IC50 values are 8.4, 39.3 and 98.3 nM respectively). PD 166285 also inhibits the checkpoint kinases Wee1 and MYT1 (Myt1), abolishes Cdc2 phosphorylation in numerous tumor cell lines, and abrogates the G2 checkpoint.西安瑞禧生物提供各種抑制劑材料。    
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